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All Publications

Synthesis of 13–epi–Taxol via a Transannular Delivery of a Borohydride Reagent
Michael Z. Hoemann, David Vander Velde, Jeffrey Aubé, Gunda I. Georg, and Lalith R. Jayasinghe
Journal of Organic Chemistry, 1995, 60, 2918–2921

https://doi.org/10.1021/jo00114a052

Structural Analysis of –Turn Mimics Containing a Substituted 6–Aminocaproic Acid Linker
Osamu Kitagawa, David Vander Velde, Dinah Dutta, Martha Morton, Fusao Takusagawa, and Jeffrey Aubé
Journal of the American Chemical Society, 1995, 117, 5169–5178

https://doi.org/10.1021/ja00124a001

Efficient Nitrogen Ring–Expansion Process Facilitated by in situ Tethering of an Alkyl Azide to Ketones. An Asymmetric Schmidt Reaction
Vijaya Gracias, Gregory L. Milligan, and Jeffrey Aubé
Journal of the American Chemical Society, 1995, 117, 8047–8048

https://doi.org/10.1021/ja00135a036

Novel Cytotoxic 3'–(tert–Butyl)–3'–dephenyl Analogs of Paclitaxel and Docetaxel
Syed M. Ali, Michael Z. Hoemann, Jeffrey Aubé, Lester A. Mitscher, Gunda I. Georg, Randy McCall, and Lalith R. Jayasinghe
Journal of Medicinal Chemistry, 1995, 38, 3821–3828

https://doi.org/10.1021/jm00019a012

Intramolecular Schmidt Reactions of Alkyl Azides with Ketones: Scope and Stereochemical Studies
Gregory L. Milligan, Craig J. Mossman, and Jeffrey Aubé
Journal of the American Chemical Society, 1995, 117, 10449–10459

https://doi.org/10.1021/ja00147a006

Conformational Analysis and Structural Elucidation of Spirocyclic Oxaziridines Using NMR, Crystallography, and Molecular Modeling
Yoshinosuke Usuki, Yuguang Wang, and Jeffrey Aubé
Journal of Organic Chemistry, 1995, 60, 8028–8035

https://doi.org/10.1021/jo00129a050

N-(tert-Butoxycarbonyloxy)phthalimide
Michael S. Wolfe and Jeffrey Aubé
John Wiley and Sons: Sussex, 1995; Volume 2, pp. 838-839.

Synthesis of Functionalized N–Alkyl Heterocycles from Ketones by a Sequential Ring Expansion/Nucleophilic Addition Sequence
Vijaya Gracias, Gregory L. Milligan, and Jeffrey Aubé
Journal of Organic Chemistry, 1996, 61, 10–11

https://doi.org/10.1021/jo951953w

Total Synthesis of Curacin A
Michael Z. Hoemann, Konstantinos A. Agrios, and Jeffrey Aubé
Tetrahedron Letters, 1996, 37, 953–956

https://doi.org/10.1016/0040-4039(95)02337-2

Asymmetric Approaches to the Yohimbine Alkaloids: Development of a Group-Selective Ring-Expansion Process and Its Application to Total Synthesis
Jeffrey Aubé and Shomir Ghosh
JAI Press: Greenwich, Connecticut, 1996, pp. 99-150.

Toward the Synthesis of Sparteine: Intramolecular Schmidt Reactions on a Norbornanone Platform
John A. Wendt and Jeffrey Aubé
Tetrahedron Letters, 1996, 37, 1531–1534

https://doi.org/10.1016/0040-4039(96)00100-1

Intramolecular Schmidt Reactions of Alkyl Azides with Ketals and Enol Ethers
Craig J. Mossman and Jeffrey Aubé
Tetrahedron, 1996, 52, 3403–3408

https://doi.org/10.1016/0040-4020(96)00037-3

Principles of Asymmetric Synthesis
Robert E. Gawley and Jeffrey Aubé
Pergamon Press: Oxford, 1996, 372 pp.

One–Step Conversion of Aldehydes to Oxazolines and 5,6–Dihydro–4H–[1,3]–oxazines Using 1,2– and 1,3–Azido Alcohols
Jennifer G. Badiang and Jeffrey Aubé
Journal of Organic Chemistry, 1996, 61, 2484–2487

https://doi.org/10.1021/jo9521256

Butitaxel Analogues: Synthesis and Structure–Activity Relationships
Syed M. Ali, Michael Z. Hoemann, Jeffrey Aubé, Gunda I. Georg, Lester A. Mitscher, and Lalith R. Jayasinghe
Journal of Medicinal Chemistry, 1997, 40, 236–241

https://doi.org/10.1021/jm960505t

Stereoselective Synthesis of Freidinger Lactams Using Oxaziridines Derived from Amino Acids
Michael S. Wolfe, Dinah Dutta, and Jeffrey Aubé
Journal of Organic Chemistry, 1997, 62, 654–663

https://doi.org/10.1021/jo961670j

Total Synthesis of (+)–Curacin A, a Marine Cytotoxic Agent
Michael Z. Hoemann, Konstantinos A. Agrios, and Jeffrey Aubé
Tetrahedron, 1997, 53, 11087–11098

https://doi.org/10.1016/S0040-4020(97)00368-2

Improvement of Oral Peptide Bioavailability: Peptidomimetic and Prodrug Strategies
Giovanni M. Pauletti, Sankeev Gangwar, Teruna J. Siaahan, Jeffrey Aubé, and Ronald T. Borchardt
Advanced Drug Delivery Reviews, 1997, 27, 235-256

https://doi.org/10.1016/S0169-409X(97)00045-8

Oxaziridine Rearrangements in Asymmetric Synthesis
Jeffrey Aubé
Chemical Society Reviews, 1997, 26, 269-277

https://doi.org/10.1039/CS9972600269

Effect of Stereochemistry on the Transport of Aca–Linked –Turn Peptidomimetics Across a Human Intestinal Cell Line
Kiyoshi Tamura, Konstantinos A. Agrios, David Vander Velde, Jeffrey Aubé, and Ronald T. Borchardt
Bioorganic and Medicinal Chemistry, 1997, 5, 1859–1866

https://doi.org/10.1016/S0968-0896(97)00115-6

Ring Expansion by in situ Tethering of Hydroxy Azides to Ketones: The Boyer Reaction
Vijaya Gracias, Kristine E. Frank, Gregory L. Milligan, and Jeffrey Aubé
Tetrahedron, 1997, 53, 16241–16252

https://doi.org/10.1016/S0040-4020(97)01012-0

Asymmetric Synthesis
Jeffrey Aubé
Volume 1; Macmillan Reference USA, Simon & Schuster Macmillan: New York, 1997, pp. 176-179

Synthesis of Lactam Peptidomimetics
Jeffrey Aubé
JAI Press: Greenwich, Connecticut, 1997, 193-232

Syntheses and Evaluation of Peptidyl Michael Acceptors That Inactivate Human Rhinovirus 3C Protease and Inhibit Virus Replication
Jian–she Kong, Shankar Venkatraman, Kelly Furness, Sanjay Nimkar, Timothy A. Shepard, Q. May Wang, Jeffrey Aubé, and Robert P. Hanzlik
Journal of Medicinal Chemistry, 1998, 41, 2579–2587

https://doi.org/10.1021/jm980114+

Lewis Acid–mediated Cyclizations of (2'-Amino-N'-tert-butoxycarbonylbenzylidene)-3-alkenylamines
Kristine E. Frank and Jeffrey Aubé
Tetrahedron Letters, 1998, 39, 7239–7242

https://doi.org/10.1016/S0040-4039(98)01596-2

Mannich Reactions Using Benzyl Azide as a Latent N-(Phenylamino)methylating Agent
Klaas Schildknegt, Konstantinos A. Agrios, and Jeffrey Aubé
Tetrahedron Letters, 1998, 39, 7687–7690

https://doi.org/10.1016/S0040-4039(98)01721-3

Reactions of Oxazolinium and Dihydrooxazinium Salts Prepared by an Azide Insertion Sequence: pH Control of Product Distribution
Jennifer E. Forsee, Brent T. Smith, Kristine E. Frank, and Jeffrey Aubé
Synlett, 1998, 1258–1260

https://doi.org/10.1055/s-1998-1925

Design, Synthesis and Evaluation of Azapeptides as Substrates and Inhibitors for Human Rhinovirus 3C Protease
Shankar Venkatraman, Jian-she Kong, Sanjay Nimkar, Q. May Wang, Jeffrey Aubé, and Robert P. Hanzlik
Bioorganic and Medicinal Chemistry Letters, 1999, 9, 577–580

https://doi.org/10.1016/S0960-894X(99)00049-9

Hydrolysis of Iminium Ethers Derived from the Reaction of Ketones with Hydroxy Azides:  Synthesis of Macrocyclic Lactams and Lactones
Jennifer E. Forsee and Jeffrey Aubé
Journal of Organic Chemistry, 1999, 64, 4381–4385

https://doi.org/10.1021/jo990041h

1,7–Asymmetric Induction in a Nitrogen Ring Expansion Process Facilitated by in situ Tethering
Kelly Furness and Jeffrey Aubé
Organic Letters, 1999, 1, 495–497

https://doi.org/10.1021/ol990685b

Publications

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