All Publications

Synthesis of 13–epi–Taxol via a Transannular Delivery of a Borohydride Reagent
Michael Z. Hoemann, David Vander Velde, Jeffrey Aubé, Gunda I. Georg, and Lalith R. Jayasinghe
Journal of Organic Chemistry, 1995, 60, 2918–2921
Structural Analysis of –Turn Mimics Containing a Substituted 6–Aminocaproic Acid Linker
Osamu Kitagawa, David Vander Velde, Dinah Dutta, Martha Morton, Fusao Takusagawa, and Jeffrey Aubé
Journal of the American Chemical Society, 1995, 117, 5169–5178
Efficient Nitrogen Ring–Expansion Process Facilitated by in situ Tethering of an Alkyl Azide to Ketones. An Asymmetric Schmidt Reaction
Vijaya Gracias, Gregory L. Milligan, and Jeffrey Aubé
Journal of the American Chemical Society, 1995, 117, 8047–8048
Novel Cytotoxic 3'–(tert–Butyl)–3'–dephenyl Analogs of Paclitaxel and Docetaxel
Syed M. Ali, Michael Z. Hoemann, Jeffrey Aubé, Lester A. Mitscher, Gunda I. Georg, Randy McCall, and Lalith R. Jayasinghe
Journal of Medicinal Chemistry, 1995, 38, 3821–3828
Intramolecular Schmidt Reactions of Alkyl Azides with Ketones: Scope and Stereochemical Studies
Gregory L. Milligan, Craig J. Mossman, and Jeffrey Aubé
Journal of the American Chemical Society, 1995, 117, 10449–10459
Conformational Analysis and Structural Elucidation of Spirocyclic Oxaziridines Using NMR, Crystallography, and Molecular Modeling
Yoshinosuke Usuki, Yuguang Wang, and Jeffrey Aubé
Journal of Organic Chemistry, 1995, 60, 8028–8035
N-(tert-Butoxycarbonyloxy)phthalimide
Michael S. Wolfe and Jeffrey Aubé
John Wiley and Sons: Sussex, 1995; Volume 2, pp. 838-839.

Synthesis of Functionalized N–Alkyl Heterocycles from Ketones by a Sequential Ring Expansion/Nucleophilic Addition Sequence
Vijaya Gracias, Gregory L. Milligan, and Jeffrey Aubé
Journal of Organic Chemistry, 1996, 61, 10–11
Total Synthesis of Curacin A
Michael Z. Hoemann, Konstantinos A. Agrios, and Jeffrey Aubé
Tetrahedron Letters, 1996, 37, 953–956
Asymmetric Approaches to the Yohimbine Alkaloids: Development of a Group-Selective Ring-Expansion Process and Its Application to Total Synthesis
Jeffrey Aubé and Shomir Ghosh
JAI Press: Greenwich, Connecticut, 1996, pp. 99-150.

Toward the Synthesis of Sparteine: Intramolecular Schmidt Reactions on a Norbornanone Platform
John A. Wendt and Jeffrey Aubé
Tetrahedron Letters, 1996, 37, 1531–1534
Intramolecular Schmidt Reactions of Alkyl Azides with Ketals and Enol Ethers
Craig J. Mossman and Jeffrey Aubé
Tetrahedron, 1996, 52, 3403–3408
Principles of Asymmetric Synthesis
Robert E. Gawley and Jeffrey Aubé
Pergamon Press: Oxford, 1996, 372 pp.

One–Step Conversion of Aldehydes to Oxazolines and 5,6–Dihydro–4H–[1,3]–oxazines Using 1,2– and 1,3–Azido Alcohols
Jennifer G. Badiang and Jeffrey Aubé
Journal of Organic Chemistry, 1996, 61, 2484–2487
Butitaxel Analogues: Synthesis and Structure–Activity Relationships
Syed M. Ali, Michael Z. Hoemann, Jeffrey Aubé, Gunda I. Georg, Lester A. Mitscher, and Lalith R. Jayasinghe
Journal of Medicinal Chemistry, 1997, 40, 236–241
Stereoselective Synthesis of Freidinger Lactams Using Oxaziridines Derived from Amino Acids
Michael S. Wolfe, Dinah Dutta, and Jeffrey Aubé
Journal of Organic Chemistry, 1997, 62, 654–663
Total Synthesis of (+)–Curacin A, a Marine Cytotoxic Agent
Michael Z. Hoemann, Konstantinos A. Agrios, and Jeffrey Aubé
Tetrahedron, 1997, 53, 11087–11098
Improvement of Oral Peptide Bioavailability: Peptidomimetic and Prodrug Strategies
Giovanni M. Pauletti, Sankeev Gangwar, Teruna J. Siaahan, Jeffrey Aubé, and Ronald T. Borchardt
Advanced Drug Delivery Reviews, 1997, 27, 235-256
Oxaziridine Rearrangements in Asymmetric Synthesis
Jeffrey Aubé
Chemical Society Reviews, 1997, 26, 269-277
Effect of Stereochemistry on the Transport of Aca–Linked –Turn Peptidomimetics Across a Human Intestinal Cell Line
Kiyoshi Tamura, Konstantinos A. Agrios, David Vander Velde, Jeffrey Aubé, and Ronald T. Borchardt
Bioorganic and Medicinal Chemistry, 1997, 5, 1859–1866
Ring Expansion by in situ Tethering of Hydroxy Azides to Ketones: The Boyer Reaction
Vijaya Gracias, Kristine E. Frank, Gregory L. Milligan, and Jeffrey Aubé
Tetrahedron, 1997, 53, 16241–16252
Asymmetric Synthesis
Jeffrey Aubé
Volume 1; Macmillan Reference USA, Simon & Schuster Macmillan: New York, 1997, pp. 176-179

Synthesis of Lactam Peptidomimetics
Jeffrey Aubé
JAI Press: Greenwich, Connecticut, 1997, 193-232

Syntheses and Evaluation of Peptidyl Michael Acceptors That Inactivate Human Rhinovirus 3C Protease and Inhibit Virus Replication
Jian–she Kong, Shankar Venkatraman, Kelly Furness, Sanjay Nimkar, Timothy A. Shepard, Q. May Wang, Jeffrey Aubé, and Robert P. Hanzlik
Journal of Medicinal Chemistry, 1998, 41, 2579–2587
Lewis Acid–mediated Cyclizations of (2'-Amino-N'-tert-butoxycarbonylbenzylidene)-3-alkenylamines
Kristine E. Frank and Jeffrey Aubé
Tetrahedron Letters, 1998, 39, 7239–7242
Mannich Reactions Using Benzyl Azide as a Latent N-(Phenylamino)methylating Agent
Klaas Schildknegt, Konstantinos A. Agrios, and Jeffrey Aubé
Tetrahedron Letters, 1998, 39, 7687–7690
Reactions of Oxazolinium and Dihydrooxazinium Salts Prepared by an Azide Insertion Sequence: pH Control of Product Distribution
Jennifer E. Forsee, Brent T. Smith, Kristine E. Frank, and Jeffrey Aubé
Synlett, 1998, 1258–1260
Design, Synthesis and Evaluation of Azapeptides as Substrates and Inhibitors for Human Rhinovirus 3C Protease
Shankar Venkatraman, Jian-she Kong, Sanjay Nimkar, Q. May Wang, Jeffrey Aubé, and Robert P. Hanzlik
Bioorganic and Medicinal Chemistry Letters, 1999, 9, 577–580
Hydrolysis of Iminium Ethers Derived from the Reaction of Ketones with Hydroxy Azides:  Synthesis of Macrocyclic Lactams and Lactones
Jennifer E. Forsee and Jeffrey Aubé
Journal of Organic Chemistry, 1999, 64, 4381–4385
1,7–Asymmetric Induction in a Nitrogen Ring Expansion Process Facilitated by in situ Tethering
Kelly Furness and Jeffrey Aubé
Organic Letters, 1999, 1, 495–497

Publications