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All Publications

Cyclizations of Substituted Benzylidene–3–alkenylamines: Synthesis of the Tricyclic Core of the Martinellines

Kristine E. Frank and Jeffrey Aubé

Journal of Organic Chemistry, 2000, 65, 655–666

https://doi.org/10.1021/jo990843c

Regiocontrol in an Intramolecular Schmidt Reaction: Total Synthesis of (+)–Aspidospermidine

Rajesh Iyengar, Klaas Schildknegt, and Jeffrey Aubé

Organic Letters, 2000, 2, 1625–1627

https://doi.org/10.1021/ol005913c

Synthesis and Conformation of Gly–Gly Dipeptides Constrained with Phenylalanine–Like Aminocaproic Acid Linkers

Mary MacDonald, David Vander Velde, and Jeffrey Aubé

Organic Letters, 2000, 2, 1653–1655

https://doi.org/10.1021/ol005618s

Regiochemical Studies of the Ring–Expansion Reactions of Hydroxy Azides with Cyclic Ketones

Brenton T. Smith, Vijaya Gracias, and Jeffrey Aubé

Journal of Organic Chemistry, 2000, 65, 3771–3774

https://doi.org/10.1021/jo000056b

Reactivity Toward Deamidation of Asparagine Residues in –Turn Structures

Xie, M.; Aubé, J.; Borchardt, R. T.; Morton, M.; Topp, E. M.; Vander Velde, D.; Schowen, R. L

Journal of Peptide Research, 2000, 56, 165–171

https://doi.org/10.1034/j.1399-3011.2000.00764.x

Synthesis of –Amino–'–diazomethyl Ketones Via Ring Opening of Substituted Cyclopropanones with Alkyl Azides. A Facile Route to N–Substituted 3–Azetidinones

Pankaj Desai and Jeffrey Aubé

Organic Letters, 2000, 2, 1657–1659

https://doi.org/10.1021/ol0056628

Reactions of Alkyl Azides and Ketones as Mediated by Lewis Acids: Schmidt and Mannich Reactions Using Azide Precursors

Pankaj Desai, Klaas Schildknegt, Konstantinos A. Agrios, Craig Mossman, Gregory L. Milligan, and Jeffrey Aubé

Journal of the American Chemical Society, 2000, 122, 7226–7232

https://doi.org/10.1021/ja000490v

Stereochemistry of the Oxidation of Imines Derived from Substituted Cyclohexanones: Axial vs. Equatorial Attack and Evidence for Delivery by an Adjacent Hydroxyl Group

Yuguang Wang, Samuel Chackalamannil, and Jeffrey Aubé

Journal of Organic Chemistry, 2000, 65, 5120–5126

https://doi.org/10.1021/jo991928g

A Functional Assay for Quantitation of the Apparent Affinities of Ligands of P–Glycoprotein in Caco–2 Cells

Jinnian Gao, Osamu Murase, Richard L. Schowen, Jeffrey Aubé, and Ronald Borchardt

Pharmaceutical Research, 2001, 18, 171–177

https://doi.org/10.1023/a:1011076217118

Transport Characteristics of Peptides and Peptidomimetics: I. N–Methylated Peptides as Substrates for the Oligopeptide Transporter and P–Glycoprotein in the Intestinal Mucosa

Jinnian Gao, Masao Sudoh, Jeffrey Aubé, and Ronald T. Borchardt

Journal of Peptide Research, 2001, 57, 316–329

https://doi.org/10.1046/j.1397-002X.2001.00000.x

Transport Characteristics of Peptides and Peptidomimetics: II. Hydroxyethylamine Bioisostere–Containing Peptidomimetics as Substrates for the Oligopeptide Transporter and P–Glycoprotein in the Intestinal Mucosa

Jinnian Gao, Stephanie L. Winslow, David Vander Velde, Jeffrey Aubé, and Ronald T. Borchardt

Journal of Peptide Research, 2001, 57, 361–373

https://doi.org/10.1034/j.1399-3011.2001.00830.x

Intramolecular Reactions of Benzylic Azides with Ketones: Competition Between Schmidt and Mannich Pathways

Aaron Wrobleski and Jeffrey Aubé

Journal of Organic Chemistry, 2001, 66, 886–889

https://doi.org/10.1021/jo001367p

Approaches to Cyclic -Turn Mimetics

Mary MacDonald and Jeffrey Aubé

Current Organic Chemistry, 2001, 5, 89-111

https://doi.org/10.2174/1385272013375517

Effect of Progressive Benzyl Substitution on the Conformations of Aminocaproic Acid–Cyclized Dipeptides

Mary MacDonald, David Vander Velde, and Jeffrey Aubé

Journal of Organic Chemistry, 2001, 66, 2636–2642

https://doi.org/10.1021/jo001308b

First Asymmetric Total Synthesis of (+)–Sparteine

Brenton T. Smith, John A. Wendt, and Jeffrey Aubé

Organic Letters, 2002, 4, 2577–2579

https://doi.org/10.1021/ol026230v

Asymmetric Total Synthesis of Dendrobatid Alkaloid 251F

Aaron Wrobleski, Kiran Sahasrabudhe, and Jeffrey Aubé

Journal of the American Chemical Society, 2002, 124, 9974–9975

https://doi.org/10.1021/ja027113y

A Combined Intramolecular Diels–Alder/Intramolecular Schmidt Reaction Process: A Formal Synthesis of (±)–Stenine

Jennifer E. Golden and Jeffrey Aubé

Angewandte Chemie, International Edition, 2002, 41, 4316–4318

<a href=https://doi.org/10.1002/1521-3773(20021115)41:223.0.CO;2-U target="_blank" style="text-decoration: underline">https://doi.org/10.1002/1521-3773(20021115)41:223.0.CO;2-U

Asymmetric Schmidt Reaction of Hydroxyalkyl Azides with Ketones

Kiran Sahasrabudhe, Vijaya Gracias, Kelly Furness, Brenton T. Smith, Christopher E. Katz, D. Srinivasa Reddy, and Jeffrey Aubé

Journal of the American Chemical Society, 2003, 125, 7914–7922

https://doi.org/10.1021/ja0348896

Rearrangements of Bicyclic Nitrones to Lactams: Comparison of Photochemical and Modified Barton Conditions

Yibin Zeng, Brenton T. Smith, John Hershberger, and Jeffrey Aubé

Journal of Organic Chemistry, 2003, 68, 8065–8067

https://doi.org/10.1021/jo035004b

Lewis Acid–Mediated Reactions of Alkyl Azides with ,–Unsaturated Ketones

Srinivasa Reddy, Weston R. Judd, and Jeffrey Aubé

Organic Letters, 2003, 5, 3899–3902

https://doi.org/10.1021/ol0355130

Unusual Tethering Effects in the Schmidt Reaction of Hydroxyalkyl Azides with Ketones: Cation– and Steric Stabilization of a Pseudoaxial Phenyl Group

Christopher E. Katz and Jeffrey Aubé

Journal of the American Chemical Society, 2003, 125, 13948–13949

https://doi.org//ja0382361

Ring Expansive Routes to Quinolizidine Alkaloids: Formal Synthesis of (–)-Lasubine II

Vijaya Gracias, Yibin Zeng, Pankaj Desai, and Jeffrey Aubé

Organic Letters, 2003, 5, 4999-5001

https://doi.org/10.1021/ol035965c

Synthesis and Conformational Studies of Dipeptides Constrained by Disubstituted 3-(Aminoethoxy)Propionic Acid Linkers

D. Srinivasa Reddy, David Vander Velde, and Jeffrey Aubé

Journal of Organic Chemistry, 2004, 69, 1716-1719

https://doi.org/10.1021/jo035683q

Base-Promoted Reactions of Bridged Ketones and 1,3- and 1,4-Haloalkyl Azides: Competitive Alkylation vs. Azidation Reactions of Ketone Enolates

Lei Yao, Brenton T. Smith, and Jeffrey Aubé

Journal of Organic Chemistry, 2004, 69, 1720-1722

https://doi.org/10.1021/jo0356098

An Ab Initio Approach to Understanding the Stereoselectivity of Reactions between Hydroxyalkyl Azides and Ketones

N. Deborah Hewlett, Jeffrey Aubé, and Jennifer L. Radkiewicz-Poutsma

Journal of Organic Chemistry, 2004, 69, 3439-3446

https://doi.org/10.1021/jo035632t

Asymmetric Total Synthesis of Dendrobatid Alkaloids: Preparation of Indolizidine 251F and Its 3-Desmethyl Analogue Using an Intramolecular Schmidt Reaction Strategy

Aaron Wrobleski, Kiran Sahasrabudhe, and Jeffrey Aubé

Journal of the American Chemical Society, 2004, 126, 5475-5481

https://doi.org/10.1021/ja0320018

Domino Reactions That Combine an Azido-Schmidt Ring Expansion with the Diels-Alder Reaction

Yibin Zeng, D. Srinivasa Reddy, Erin Hirt, and Jeffrey Aubé

Organic Letters, 2004, 6, 4993–4995

https://doi.org/10.1021/ol047809r

Publications

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