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All Publications
Cyclizations of Substituted Benzylidene–3–alkenylamines: Synthesis of the Tricyclic Core of the Martinellines
Kristine E. Frank and Jeffrey Aubé
Journal of Organic Chemistry, 2000, 65, 655–666
Regiocontrol in an Intramolecular Schmidt Reaction: Total Synthesis of (+)–Aspidospermidine
Rajesh Iyengar, Klaas Schildknegt, and Jeffrey Aubé
Organic Letters, 2000, 2, 1625–1627
Synthesis and Conformation of Gly–Gly Dipeptides Constrained with Phenylalanine–Like Aminocaproic Acid Linkers
Mary MacDonald, David Vander Velde, and Jeffrey Aubé
Organic Letters, 2000, 2, 1653–1655
Regiochemical Studies of the Ring–Expansion Reactions of Hydroxy Azides with Cyclic Ketones
Brenton T. Smith, Vijaya Gracias, and Jeffrey Aubé
Journal of Organic Chemistry, 2000, 65, 3771–3774
Reactivity Toward Deamidation of Asparagine Residues in –Turn Structures
Xie, M.; Aubé, J.; Borchardt, R. T.; Morton, M.; Topp, E. M.; Vander Velde, D.; Schowen, R. L
Journal of Peptide Research, 2000, 56, 165–171
Synthesis of –Amino–'–diazomethyl Ketones Via Ring Opening of Substituted Cyclopropanones with Alkyl Azides. A Facile Route to N–Substituted 3–Azetidinones
Pankaj Desai and Jeffrey Aubé
Organic Letters, 2000, 2, 1657–1659
Reactions of Alkyl Azides and Ketones as Mediated by Lewis Acids: Schmidt and Mannich Reactions Using Azide Precursors
Pankaj Desai, Klaas Schildknegt, Konstantinos A. Agrios, Craig Mossman, Gregory L. Milligan, and Jeffrey Aubé
Journal of the American Chemical Society, 2000, 122, 7226–7232
Stereochemistry of the Oxidation of Imines Derived from Substituted Cyclohexanones: Axial vs. Equatorial Attack and Evidence for Delivery by an Adjacent Hydroxyl Group
Yuguang Wang, Samuel Chackalamannil, and Jeffrey Aubé
Journal of Organic Chemistry, 2000, 65, 5120–5126
A Functional Assay for Quantitation of the Apparent Affinities of Ligands of P–Glycoprotein in Caco–2 Cells
Jinnian Gao, Osamu Murase, Richard L. Schowen, Jeffrey Aubé, and Ronald Borchardt
Pharmaceutical Research, 2001, 18, 171–177
Transport Characteristics of Peptides and Peptidomimetics: I. N–Methylated Peptides as Substrates for the Oligopeptide Transporter and P–Glycoprotein in the Intestinal Mucosa
Jinnian Gao, Masao Sudoh, Jeffrey Aubé, and Ronald T. Borchardt
Journal of Peptide Research, 2001, 57, 316–329
Transport Characteristics of Peptides and Peptidomimetics: II. Hydroxyethylamine Bioisostere–Containing Peptidomimetics as Substrates for the Oligopeptide Transporter and P–Glycoprotein in the Intestinal Mucosa
Jinnian Gao, Stephanie L. Winslow, David Vander Velde, Jeffrey Aubé, and Ronald T. Borchardt
Journal of Peptide Research, 2001, 57, 361–373
Intramolecular Reactions of Benzylic Azides with Ketones: Competition Between Schmidt and Mannich Pathways
Aaron Wrobleski and Jeffrey Aubé
Journal of Organic Chemistry, 2001, 66, 886–889
Approaches to Cyclic -Turn Mimetics
Mary MacDonald and Jeffrey Aubé
Current Organic Chemistry, 2001, 5, 89-111
Effect of Progressive Benzyl Substitution on the Conformations of Aminocaproic Acid–Cyclized Dipeptides
Mary MacDonald, David Vander Velde, and Jeffrey Aubé
Journal of Organic Chemistry, 2001, 66, 2636–2642
First Asymmetric Total Synthesis of (+)–Sparteine
Brenton T. Smith, John A. Wendt, and Jeffrey Aubé
Organic Letters, 2002, 4, 2577–2579
Asymmetric Total Synthesis of Dendrobatid Alkaloid 251F
Aaron Wrobleski, Kiran Sahasrabudhe, and Jeffrey Aubé
Journal of the American Chemical Society, 2002, 124, 9974–9975
A Combined Intramolecular Diels–Alder/Intramolecular Schmidt Reaction Process: A Formal Synthesis of (±)–Stenine
Jennifer E. Golden and Jeffrey Aubé
Angewandte Chemie, International Edition, 2002, 41, 4316–4318
<a href=https://doi.org/10.1002/1521-3773(20021115)41:223.0.CO;2-U target="_blank" style="text-decoration: underline">https://doi.org/10.1002/1521-3773(20021115)41:223.0.CO;2-U
Asymmetric Schmidt Reaction of Hydroxyalkyl Azides with Ketones
Kiran Sahasrabudhe, Vijaya Gracias, Kelly Furness, Brenton T. Smith, Christopher E. Katz, D. Srinivasa Reddy, and Jeffrey Aubé
Journal of the American Chemical Society, 2003, 125, 7914–7922
Rearrangements of Bicyclic Nitrones to Lactams: Comparison of Photochemical and Modified Barton Conditions
Yibin Zeng, Brenton T. Smith, John Hershberger, and Jeffrey Aubé
Journal of Organic Chemistry, 2003, 68, 8065–8067
Lewis Acid–Mediated Reactions of Alkyl Azides with ,–Unsaturated Ketones
Srinivasa Reddy, Weston R. Judd, and Jeffrey Aubé
Organic Letters, 2003, 5, 3899–3902
Unusual Tethering Effects in the Schmidt Reaction of Hydroxyalkyl Azides with Ketones: Cation– and Steric Stabilization of a Pseudoaxial Phenyl Group
Christopher E. Katz and Jeffrey Aubé
Journal of the American Chemical Society, 2003, 125, 13948–13949
Ring Expansive Routes to Quinolizidine Alkaloids: Formal Synthesis of (–)-Lasubine II
Vijaya Gracias, Yibin Zeng, Pankaj Desai, and Jeffrey Aubé
Organic Letters, 2003, 5, 4999-5001
Synthesis and Conformational Studies of Dipeptides Constrained by Disubstituted 3-(Aminoethoxy)Propionic Acid Linkers
D. Srinivasa Reddy, David Vander Velde, and Jeffrey Aubé
Journal of Organic Chemistry, 2004, 69, 1716-1719
Base-Promoted Reactions of Bridged Ketones and 1,3- and 1,4-Haloalkyl Azides: Competitive Alkylation vs. Azidation Reactions of Ketone Enolates
Lei Yao, Brenton T. Smith, and Jeffrey Aubé
Journal of Organic Chemistry, 2004, 69, 1720-1722
An Ab Initio Approach to Understanding the Stereoselectivity of Reactions between Hydroxyalkyl Azides and Ketones
N. Deborah Hewlett, Jeffrey Aubé, and Jennifer L. Radkiewicz-Poutsma
Journal of Organic Chemistry, 2004, 69, 3439-3446
Asymmetric Total Synthesis of Dendrobatid Alkaloids: Preparation of Indolizidine 251F and Its 3-Desmethyl Analogue Using an Intramolecular Schmidt Reaction Strategy
Aaron Wrobleski, Kiran Sahasrabudhe, and Jeffrey Aubé
Journal of the American Chemical Society, 2004, 126, 5475-5481
Domino Reactions That Combine an Azido-Schmidt Ring Expansion with the Diels-Alder Reaction
Yibin Zeng, D. Srinivasa Reddy, Erin Hirt, and Jeffrey Aubé
Organic Letters, 2004, 6, 4993–4995
Publications
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