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All Publications

Modular Synthesis of Cyclic Peptidomimetics Inspired by -Turns

Senthil Kumar Ramanathan, John Keeler, Huey-Lih Lee, D. Srinavasa Reddy, Gerald Lushington, and Jeffrey Aubé

Organic Letters, 2005, 7, 1059-1062

https://doi.org/10.1021/ol047323a

Facile C–N Cleavage in a Series of Bridged Lactams

Yao Lei, Aaron D. Wrobleski, Jennifer E. Golden, Douglas R. Powell, and Jeffrey Aubé

Journal of the American Chemical Society, 2005, 127, 4552-4553

https://doi.org/10.1021/ja050214m

Synthesis of a Small Library of Diketopiperazines as Potential Inhibitors of Calpain

Yibin Zeng, Qingshan Li, Robert P. Hanzlik, and Jeffrey Aubé

Bioorganic and Medicinal Chemistry Letters, 2005, 15, 3034–3038

https://doi.org/10.1016/j.bmcl.2005.04.031

Regioselective Single and Double Conjugate Additions to Substituted Cyclohexa-2,5-Dienone Monoacetals

Scott Grecian, Aaron D. Wrobleski, and Jeffrey Aubé

Organic Letters, 2005, 7, 3167–3170

https://doi.org/10.1021/ol050715c

Amides and Derivatives; Polyamides and Peptides: Lactams. 21.1.5. Product Subclass 1: Synthesis by Rearrangement

Weston Judd, Christopher E. Katz, and Jeffrey Aubé

George Thieme Verlag KG: Stuttgart, 2005, 133–178

An Expeditious Total Synthesis of (±)-Stenine

Yibin Zeng and Jeffrey Aubé

Journal of the American Chemical Society, 2005, 127, 15712–15713

https://doi.org/10.1021/ja055629m

Revisiting a Classic Approach to the Aspidosperma Alkaloids: An Intramolecular Schmidt Reaction-Mediated Synthesis of (+)-Aspidospermidine

Rajesh Iyengar, Klaas Schildknegt, Martha Morton, and Jeffrey Aubé

Journal of Organic Chemistry, 2005, 70, 10645-10662

https://doi.org/10.1021/jo051212n

Cyclization of a Carbon-Centered Radical Derived from Oxaziridine Cleavage

Yoshinosuke Usuki, Xin Peng, Belgin Gülgeze, and Jeffrey Aubé

Arkivoc, 2006, part iv, 189–199

https://doi.org/10.3998/ark.5550190.0007.413

Remote Control of Diastereoselectivity in Intramolecular Reactions of Chiral Allylsilanes

Weston R. Judd, Sooho Ban, and Jeffrey Aubé

Journal of the American Chemical Society, 2006, 128, 13736–13741

https://doi.org/10.1021/ja063411+

Solution-Phase Parallel Synthesis of a Library of 2-Pyrazolines

Shankar Manyem, Mukund P. Sibi, Gerald H. Lushington, Benjamin Neuenswander, Frank Schoenen, and Jeffrey Aubé

Journal of Combinatorial Chemistry, 2007, 9, 20–28

https://doi.org/10.1021/cc0601175

Cation– Control of Regiochemistry of Intramolecular Schmidt Reactions en Route to Bridged Bicyclic Lactams

Lei Yao and Jeffrey Aubé

Journal of the American Chemical Society, 2007, 129, 2766–2767

https://doi.org/10.1021/ja068919r

One-Step Synthesis of Oxazoline and Dihydrooxazine Libraries

Priyanka Chaudhry, Frank Schoenen, Benjamin Neuenswander, Gerald H. Lushington, and Jeffrey Aubé

Journal of Combinatorial Chemistry, 2007, 9, 473–476

https://doi.org/10.1021/cc060159t

Intramolecular and Intermolecular Schmidt Reactions of Alkyl Azides with Aldehydes

Huey-Lih Lee and Jeffrey Aubé

Tetrahedron, 2007, 63, 9007–9015

https://doi.org/10.1016/j.tet.2007.05.079

Synthesis of an N-Substituted Lactam Using an Intramolecular Schmidt Reaction

Scott Grecian and Jeffrey Aubé

Organic Syntheses, 2007, 84, 347–358

https://doi.org/10.15227/orgsyn.084.0347

Double Conjugate Addition of a Nitropropionate Ester to a Quinone Monoketal: Synthesis of an Advanced Intermediate to (±)-Gelsemine

Scott Grecian and Jeffrey Aubé

Organic Letters, 2007, 9, 3153–3156

https://doi.org/10.1021/ol071174p

Synthesis of Isoquinol-1-one-8-carboxylic Acid Libraries Using a Tandem Diels–Alder/Acylation Sequence

Kevin J. Frankowski, Erin E. Hirt, Yibin Zeng, Ben Neuenswander, Drew Fowler, Frank Schoenen, and Jeffrey Aubé

Journal of Combinatorial Chemistry, 2007, 9, 1188–1192

https://doi.org/10.1021/cc700127f

Reactions of Cyclopropanone Acetals with Alkyl Azides: Carbonyl Addition versus Ring-Opening Pathways

Scott Grecian, Pankaj Desai, Craig Mossman, Jennifer L. Poutsma, and Jeffrey Aubé

Journal of Organic Chemistry, 2007, 72, 9439–9447

https://doi.org/10.1021/jo0711034

Nucleophilic Addition to Iminium Ethers in the Preparation of Functionalized N-Alkyl Heterocycles

Erik Fenster, Brenton T. Smith, Vijaya Gracias, Gregory L. Milligan, and Jeffrey Aubé

Journal of Organic Chemistry, 2008, 73, 201–205

https://doi.org/10.1021/jo702193g

Synthesis of Enantiomerically Enriched (R)-5-tert-Butylazepan-2-one Using a Hydroxyalkyl-azide Mediated Ring Expansion Reaction

Timothy P. Ribelin and Jeffrey Aubé

Nature: Protocols, 2008, 3, 137–143

https://doi.org/10.1038/nprot.2007.518

Three-Component Synthesis of 1,4-Diazepin-5-ones and the Construction of γ Turn-like Peptidomimetic Libraries

Erik Fenster, Dinesh K. Rayabarapu, Mianji Zhang, Shubhasish Mukherjee, David Hill, Ben Neuenswander, Frank Schoenen, Paul R. Hanson, and Jeffrey Aubé

Journal of Combinatorial Chemistry, 2008, 10, 230–234

https://doi.org/10.1021/cc700174c

Efficient Synthesis of γ-Lactams by a Tandem Reductive Amination/Lactamization Sequence

Julica Nöth, Kevin J. Frankowski, Benjamin Neuenswander, Jeffrey Aubé, and Oliver Reiser

Journal of Combinatorial Chemistry, 2008, 10, 456–459

https://doi.org/10.1021/cc700202c

Syntheses of the Stemona Alkaloids (±)-Stenine, (±)-Neostenine, and (±)-13-Epineostenine Using a Stereodivergent Diels–Alder/Azido-Schmidt Reaction

Kevin J. Frankowski, Jennifer E. Golden, Yibin Zeng, Yao Lei, and Jeffrey Aubé

Journal of the American Chemical Society, 2008, 130, 6018–6024

https://doi.org/10.1021/ja800574m

Non-Bonded, Attractive Cation– Interactions in Azide-Mediated Asymmetric Ring Expansion Reactions

Christopher E. Katz, Timothy Ribelin, Donna Withrow, Yashar Basseri, Anna K. Manukyan, Amy Bermudez, Christian G. Nuera, Victor W. Day, Douglas R. Powell, Jennifer L. Poutsma, and Jeffrey Aubé

Journal of Organic Chemistry, 2008, 73, 3318 - 3327

https://doi.org/10.1021/jo800222r

Highly Stereoselective Ring Expansion Reactions Mediated by Attractive, Non-Bonded Cation–n Interactions

Timothy Ribelin, Christopher E. Katz, Donna G. English, Sherriel Smith, Anna Manukyan, Victor W. Day, Benjamin Neuenswander, Jennifer L. Poutsma, and Jeffrey Aubé

Angewandte Chemie, International Edition, 2008, 47, 6233–6235

https://doi.org/10.1002/anie.200801591

Explorations of Stemona Alkaloid-Inspired Analogues: Skeletal Modification and Functional Group Diversification

Kevin J. Frankowski, Benjamin Neuenswander, and Jeffrey Aubé

Journal of Combinatorial Chemistry, 2008, 10, 721-725

https://doi.org/10.1021/cc800078h

The Total Synthesis of Amphibian Alkaloids Using the Intramolecular Schmidt Reaction

Kevin J. Frankowski, Aaron Wrobleski and Jeffrey Aubé,

Elsevier: Amsterdam, 2008, 408–459

Synthesis and Structural Study of Cyclic 5-Aminovaleric Acid-linked -Ala–-Ala Dipeptides

Anne Mengel, Oliver Reiser, and Jeffrey Aubé

Bioorganic & Medicinal Chemistry Letters, 2008, 18, 5975-5977

https://doi.org/10.1016/j.bmcl.2008.07.082

Stability of Medium-Bridged Twisted Amides in Aqueous Solutions

Michal Szostak, Lei Yao, and Jeffrey Aubé

Journal of Organic Chemistry, 2009, 74, 1869–1875

https://doi.org/10.1021/jo802192v

“Direct Synthesis of Medium-Bridged Twisted Amides via a Transannular Cyclization Strategy

Michal Szostak and Jeffrey Aubé

Organic Letters, 2009, 11, 3878–3881

https://doi.org/10.1021/ol901449y

Asymmetric Total Synthesis of Alkaloids 223A and 6-epi-223A

Partha Ghosh, Weston R. Judd, Timothy Ribelin, and Jeffrey Aubé

Organic Letters, 2009, 11, 4140–4142

https://doi.org/10.1021/ol901645j

Corey–Chaykovsky Epoxidation of Twisted Amides: Synthesis and Reactivity of Bridged Spiro-epoxyamines

Michal Szostak and Jeffrey Aubé

Journal of the American Chemical Society, 2009, 131, 13246–13247

https://doi.org/10.1021/ja906471q

Schmidt Rearrangement Reactions with Alkyl Azides

Scott Grecian and Jeffrey Aubé

John Wiley and Sons: Chichester, UK, 2009, pp 191-237

Cation−n Control of Regiochemistry of Intramolecular Schmidt Reactions en Route to Bridged Bicyclic Lactams

Michal Szostak, Lei Yao, and Jeffrey Aubé

Organic Letters, 2009, 11, pp 4386–4389

https://doi.org/10.1021/ol901771b

One-pot Synthesis of Lactams Using Domino Reactions: Combination of Schmidt Reaction with Sakurai and Aldol Reactions

Chan Woo Huh, Gagandeep K. Somal, Christopher E. Katz, Huaxing Pei, Yibin Zeng, Justin T. Douglas, and Jeffrey Aubé

Journal of Organic Chemistry, 2009, 74, 7618–7626

https://doi.org/10.1021/jo901843w

Synthesis and Rearrangement of a Bridged Thioamide

Michal Szostak and Jeffrey Aubé

Chemical Communications, 2009, 7122–7124

https://doi.org/10.1039/b917508c

Publications

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